SbCl3 as an Efficient Catalyst for the One-pot Synthesis of Highly Substituted Piperidines

Authors

  • Malek Taher Maghsoodlou* Department of Chemistry, Faculty of Science, University of Sistan and Baluchestan, P. O. Box: 98135-674, Zahedan, Iran
Abstract:

Highly substituted piperidines were synthesized via the condensation of aromatic aldehydes and aromatic amines with β-ketoesters in the presence of antimony(III) chloride at ambient condition. This reaction has any advantages such as easy work-up, clean procedure, and good yields.

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Journal title

volume 3  issue 2

pages  119- 125

publication date 2017-10-01

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